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2019

Leveraging a Low-Affinity Diazaspiro Orthosteric Fragment to Reduce Dopamine D 3 Receptor (D 3 R) Ligand Promiscuity across Highly Conserved Aminergic G-Protein-Coupled Receptors (GPCRs)

Reilly, S. W., Riad, A. A., Hsieh, C. J., Sahlholm, K., Jacome, D. A., Griffin, S., Taylor, M., Weng, C. C., Xu, K., Kirschner, N., Luedtke, R. T., Parry, C., Malhotra, S., Karanicolas, J. & Mach, R. H., 23 May 2019, In : Journal of Medicinal Chemistry. 62, 10, p. 5132-5147 16 p.

Research output: Contribution to journalArticleResearchpeer-review

G-Protein-Coupled Receptors
Dopamine
Ligands
Adrenergic Agents
Pharmaceutical Preparations

Retraction notice to “Dopamine Ds3 receptor partial agonist LS-3-134 attenuates cocaine-motivated behaviors” [Pharmacology, Biochemistry and Behavior 171 (2018) 46–53](S0091305718300236)(10.1016/j.pbb.2018.05.015)

Powell, G. L., Bonadonna, J. P., Vannan, A., Xu, K., Mach, R. H., Luedtke, R. T. & Neisewander, J. L., 1 Jan 2019, In : Pharmacology Biochemistry and Behavior. 176, 1 p.

Research output: Contribution to journalComment/debateResearch

Biochemistry
Dopamine Receptors
Cocaine
Animal Care Committees
Pharmacology
2018
1 Citation (Scopus)

Analogues of Arylamide Phenylpiperazine Ligands to Investigate the Factors Influencing D3 Dopamine Receptor Bitropic Binding and Receptor Subtype Selectivity

Hayatshahi, H. S., Xu, K., Griffin, S. A., Taylor, M., Mach, R. H., Liu, J. & Luedtke, R. T., 19 Dec 2018, In : ACS Chemical Neuroscience. 9, 12, p. 2972-2983 12 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Ligands
Dopamine D2 Receptors
Dopamine Receptors
Nitrogen
6 Citations (Scopus)

Challenges in the development of dopamine D2- and D3-selective radiotracers for PET imaging studies

Mach, R. H. & Luedtke, R. T., 1 Mar 2018, In : Journal of Labelled Compounds and Radiopharmaceuticals. 61, 3, p. 291-298 8 p.

Research output: Contribution to journalArticleResearchpeer-review

Positron emission tomography
Positron-Emission Tomography
Dopamine D2 Receptors
Dopamine
Dopamine D3 Receptors
12 Citations (Scopus)

Dissociation of striatal dopamine and tyrosine hydroxylase expression from aging-related motor decline: Evidence from calorie restriction intervention

Salvatore, M. F., Terrebonne, J., Cantu, M. A., McInnis, T. R., Venable, K., Kelley, P., Kasanga, E. A., Latimer, B., Owens, C. L., Pruett, B. S., Yu, Y., Luedtke, R. T., Forster, M. J., Sumien, N. & Ingram, D. K., 1 Jan 2018, In : Journals of Gerontology - Series A Biological Sciences and Medical Sciences. 73, 1, p. 11-20 10 p.

Research output: Contribution to journalArticleResearchpeer-review

Corpus Striatum
Tyrosine 3-Monooxygenase
Dopamine
Locomotion
Hypokinesia

Dopamine D3 receptor partial agonist LS-3-134 attenuates cocaine-motivated behaviors

Powell, G. L., Bonadonna, J. P., Vannan, A., Xu, K., Mach, R. H., Luedtke, R. T. & Neisewander, J. L., 1 Dec 2018, In : Pharmacology Biochemistry and Behavior. 175, p. 123-129 7 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Cocaine
Reinforcement Schedule
Reinforcement
Locomotion

Dopamine D3 receptor partial agonist LS-3-134 attenuates cocaine-motivated behaviors

Powell, G. L., Bonadonna, J. P., Vannan, A., Xu, K., Mach, R. H., Luedtke, R. T. & Neisewander, J. L., 1 Aug 2018, In : Pharmacology Biochemistry and Behavior. 171, p. 46-53 8 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Cocaine
Reinforcement Schedule
Reinforcement
Locomotion
2017

Dysregulated corticostriatal activity in open-field behavior and the head-twitch response induced by the hallucinogen 2,5-dimethoxy-4-iodoamphetamine

Rangel-Barajas, C., Estrada-Sánchez, A. M., Barton, S. J., Luedtke, R. T. & Rebec, G. V., 1 Feb 2017, In : Neuropharmacology. 113, p. 502-510 9 p.

Research output: Contribution to journalArticleResearchpeer-review

Hallucinogens
Head
Neurons
Motor Cortex
Amphetamine
3 Citations (Scopus)

Highly Selective Dopamine D3 Receptor Antagonists with Arylated Diazaspiro Alkane Cores

Reilly, S. W., Griffin, S., Taylor, M., Sahlholm, K., Weng, C. C., Xu, K., Jacome, D. A., Luedtke, R. T. & Mach, R. H., 14 Dec 2017, In : Journal of Medicinal Chemistry. 60, 23, p. 9905-9910 6 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Alkanes
Dopamine Antagonists
Ligands
2016
1 Citation (Scopus)

The effect of the sigma-1 receptor selective compound LS-1-137 on the DOI-induced head twitch response in mice

Malik, M., Rangel-Barajas, C., Mach, R. H. & Luedtke, R. T., 1 Sep 2016, In : Pharmacology Biochemistry and Behavior. 148, p. 136-144 9 p.

Research output: Contribution to journalArticleResearchpeer-review

Head
Receptor, Serotonin, 5-HT2C
sigma Receptors
sigma-1 receptor
N-(1-benzylpiperidin-4-yl)phenylacetamide
2015
7 Citations (Scopus)

Bitropic D3 dopamine receptor selective compounds as potential antipsychotics

Luedtke, R. T., Rangel-Barajas, C., Malik, M., Reichert, D. E. & Mach, R. H., 1 Sep 2015, In : Current Pharmaceutical Design. 21, 26, p. 3700-3724 25 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Antipsychotic Agents
Dopamine D2 Receptors
Dopamine D4 Receptors
Ligands
5 Citations (Scopus)

Pharmacological modulation of abnormal involuntary DOI-induced head twitch response movements in male DBA/2J mice: II. Effects of D3 dopamine receptor selective compounds

Rangel-Barajas, C., Malik, M., Mach, R. H. & Luedtke, R. T., 1 Jan 2015, In : Neuropharmacology. 93, p. 179-190 12 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Inbred DBA Mouse
Head
Pharmacology
Dopamine D2 Receptors
6 Citations (Scopus)

Synthesis, pharmacological evaluation and molecular modeling studies of triazole containing dopamine D 3 receptor ligands

Peng, X., Wang, Q., Mishra, Y., Xu, J., Reichert, D. E., Malik, M., Taylor, M., Luedtke, R. T. & Mach, R. H., 1 Feb 2015, In : Bioorganic and Medicinal Chemistry Letters. 25, 3, p. 519-523 5 p.

Research output: Contribution to journalArticleResearchpeer-review

Triazoles
Molecular modeling
Dopamine
Pharmacology
Ligands
16 Citations (Scopus)

The effects of sigma (σ1) receptor-selective ligands on muscarinic receptor antagonist-induced cognitive deficits in mice

Malik, M., Rangel-Barajas, C., Sumien, N., Su, C., Singh, M., Chen, Z., Huang, R-Q., Meunier, J., Maurice, T., Mach, R. H. & Luedtke, R. T., 1 May 2015, In : British Journal of Pharmacology. 172, 10, p. 2519-2531 13 p.

Research output: Contribution to journalArticleResearchpeer-review

Muscarinic Antagonists
Muscarinic Receptors
Ligands
Scopolamine Hydrobromide
Nootropic Agents
2014
10 Citations (Scopus)

Characterization of [3H]LS-3-134, a novel arylamide phenylpiperazine D3 dopamine receptor selective radioligand

Rangel-Barajas, C., Malik, M., Taylor, M., Neve, K. A., Mach, R. H. & Luedtke, R. T., 1 Nov 2014, In : Journal of Neurochemistry. 131, 4, p. 418-431 14 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Dopamine D2 Receptors
Rats
Competitive Binding
Caudate Nucleus
24 Citations (Scopus)

Design, synthesis, and structure-activity relationship studies of a series of [4-(4-carboxamidobutyl)]-1-arylpiperazines: Insights into structural features contributing to dopamine D3 versus D2 receptor subtype selectivity

Ananthan, S., Saini, S. K., Zhou, G., Hobrath, J. V., Padmalayam, I., Zhai, L., Bostwick, J. R., Antonio, T., Reith, M. E. A., McDowell, S., Cho, E., McAleer, L., Taylor, M. & Luedtke, R. T., 1 Jan 2014, In : Journal of Medicinal Chemistry. 57, 16, p. 7042-7060 19 p.

Research output: Contribution to journalArticleResearchpeer-review

Structure-Activity Relationship
Dopamine
Dopamine D3 Receptors
Ligands
Dopamine D2 Receptors
11 Citations (Scopus)

Pharmacological modulation of abnormal involuntary DOI-induced head twitch response in male DBA/2J mice: I. Effects of D2/D3 and D2 dopamine receptor selective compounds

Rangel-Barajas, C., Malik, M., Vangveravong, S., Mach, R. H. & Luedtke, R. T., 1 Jan 2014, In : Neuropharmacology. 83, p. 18-27 10 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Inbred DBA Mouse
Dopamine D2 Receptors
Head
Pharmacology
2013

Drug Design for Addiction - Molecular Determinants of Selectivity and Efficacy at the Dopamine D3 Receptor

Newman, A. H., Banala, A. K., Donthamsetti, P., Cao, J., Michino, M., Luedtke, R. T., Javitch, J. A. & Shi, L., 1 Dec 2013, Catecholamine Research in the 21st Century: Abstracts and Graphical Abstracts, 10th International Catecholamine Symposium, 2012. Elsevier Inc., p. 181-182 2 p.

Research output: Chapter in Book/Report/Conference proceedingChapterResearchpeer-review

Dopamine D3 Receptors
Drug Design
Substance-Related Disorders
7 Citations (Scopus)

Evaluation of N-phenyl homopiperazine analogs as potential dopamine D 3 receptor selective ligands

Li, A., Mishra, Y., Malik, M., Wang, Q., Li, S., Taylor, M., Reichert, D. E., Luedtke, R. T. & MacH, R. H., 1 Jun 2013, In : Bioorganic and Medicinal Chemistry. 21, 11, p. 2988-2998 11 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Assays
Dopamine
Dopamine D2 Receptors
Ligands
2 Citations (Scopus)

Fos expression in response to dopamine d3-preferring phenylpiperazine drugs given with and without cocaine

Nolan, B. C., Liu, S., Hammerslag, L. R., Cheung, T. H. C., Lenz, J., Mach, R. H., Luedtke, R. T. & Neisewander, J. L., 1 Dec 2013, In : Synapse. 67, 12, p. 847-855 9 p.

Research output: Contribution to journalArticleResearchpeer-review

Cocaine
Dopamine
Adenylyl Cyclases
Pharmaceutical Preparations
Nucleus Accumbens
17 Citations (Scopus)

Reduction of cocaine self-administration and D3 receptor-mediated behavior by two novel dopamine D3 receptor-selective partial agonists, OS-3-106 and WW-III-55

Cheung, T. H. C., Loriaux, A. L., Weber, S. M., Chandler, K. N., Lenz, J. D., Schaan, R. F., Mach, R. H., Luedtke, R. T. & Neisewander, J. L., 1 Nov 2013, In : Journal of Pharmacology and Experimental Therapeutics. 347, 2, p. 410-423 14 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Self Administration
Cocaine
Yawning
Sucrose
1 Citation (Scopus)

Synthesis and in vitro pharmacological evaluation of indolyl carboxylic amide analogues as D3 dopamine receptor selective ligands

Tu, Z., Li, S., Li, A., Taylor, M., Ho, D., Malik, M., Luedtke, R. T. & Mach, R. H., 1 Jan 2013, In : MedChemComm. 4, 9, p. 1283-1289 7 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Amides
Pharmacology
Ligands
Colforsin
2 Citations (Scopus)

The effect of SV 293, a D2 dopamine receptor-selective antagonist, on D2 receptor-mediated GIRK channel activation and adenylyl cyclase inhibition

Huang, R-Q., Griffin, S. A., Taylor, M., Vangveravong, S., Mach, R. H., Dillon, G. H. & Luedtke, R. T., 1 Jan 2013, In : Pharmacology. 92, 1-2, p. 84-89 6 p.

Research output: Contribution to journalArticleResearchpeer-review

Adenylyl Cyclases
Dopamine D2 Receptors
G Protein-Coupled Inwardly-Rectifying Potassium Channels
Dopamine D4 Receptors
Dopamine D3 Receptors
2012
23 Citations (Scopus)

Comparison of the binding and functional properties of two structurally different D2 dopamine receptor subtype selective compounds

Luedtke, R. T., Mishra, Y., Wang, Q., Griffin, S. A., Bell-Horner, C., Taylor, M., Vangveravong, S., Dillon, G. H., Huang, R-Q., Reichert, D. E. & MacH, R. H., 19 Dec 2012, In : ACS Chemical Neuroscience. 3, 12, p. 1050-1062 13 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Dopamine D2 Receptors
Assays
Adenylyl Cyclases
G Protein-Coupled Inwardly-Rectifying Potassium Channels
35 Citations (Scopus)

Endothelin b receptors contribute to retinal ganglion cell loss in a rat model of glaucoma

Minton, A. Z., Phatak, N. R., Stankowska, D. L., He, S., Ma, H. Y., Mueller, B. H., Jiang, M., Luedtke, R. T., Yang, S., Brownlee, C. & Krishnamoorthy, R., 20 Aug 2012, In : PLoS ONE. 7, 8, e43199.

Research output: Contribution to journalArticleResearchpeer-review

Endothelin Receptors
glaucoma
endothelins
Retinal Ganglion Cells
Endothelins

Erratum: Influence of cocaine history on the behavioral effects of dopamine d3 receptor-selective compounds in monkeys (Neuropsychopharmacology (2011) 36 (1104-1113) DOI: 10.1038/npp.2010.248)

Blaylock, B. L., Gould, R. W., Banala, A., Grundt, P., Luedtke, R. T., Newman, A. H. & Nader, M. A., 1 Oct 2012, In : Neuropsychopharmacology. 37, 11, 1 p.

Research output: Contribution to journalComment/debateResearch

Dopamine D3 Receptors
Cocaine
Haplorhini
History
96 Citations (Scopus)

Molecular determinants of selectivity and efficacy at the dopamine D3 receptor

Newman, A. H., Beuming, T., Banala, A. K., Donthamsetti, P., Pongetti, K., Labounty, A., Levy, B., Cao, J., Michino, M., Luedtke, R. T., Javitch, J. A. & Shi, L., 9 Aug 2012, In : Journal of Medicinal Chemistry. 55, 15, p. 6689-6699 11 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Binding Sites
Ligands
Sequence Homology
Substance-Related Disorders
17 Citations (Scopus)

Neuroprotective effects of high affinity sigma 1 receptor selective compounds

Luedtke, R. T., Perez, E., Yang, S., Liu, R., Vangveravong, S., Tu, Z., MacH, R. H. & Simpkins, J. W., 2 Mar 2012, In : Brain Research. 1441, p. 17-26 10 p.

Research output: Contribution to journalArticleResearchpeer-review

Neuroprotective Agents
Haloperidol
Stroke
sigma Receptors
Pentazocine
16 Citations (Scopus)

Phenylpiperazine derivatives with selectivity for dopamine D3 receptors modulate cocaine self-administration in rats

Cheung, T. H. C., Nolan, B. C., Hammerslag, L. R., Weber, S. M., Durbin, J. P., Peartree, N. A., MacH, R. H., Luedtke, R. T. & Neisewander, J. L., 1 Dec 2012, In : Neuropharmacology. 63, 8, p. 1346-1359 14 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Self Administration
Cocaine
Sucrose
Locomotion
2011
27 Citations (Scopus)

Decreased striatal dopamine receptor binding in primary focal dystonia: A D2 or D3 defect?

Karimi, M., Moerlein, S. M., Videen, T. O., Luedtke, R. T., Taylor, M., Mach, R. H. & Perlmutter, J. S., 1 Jan 2011, In : Movement Disorders. 26, 1, p. 100-106 7 p.

Research output: Contribution to journalArticleResearchpeer-review

Benperidol
Dystonic Disorders
Corpus Striatum
Dystonia
Dopamine Receptors
7 Citations (Scopus)

Effect of cyclosporin A on the uptake of D3-selective PET radiotracers in rat brain

Tu, Z., Li, S., Xu, J., Chu, W., Jones, L. A., Luedtke, R. R. & Mach, R. H., 1 Jul 2011, In : Nuclear Medicine and Biology. 38, 5, p. 725-739 15 p.

Research output: Contribution to journalArticleResearchpeer-review

Cyclosporine
Electrons
Brain
ATP-Binding Cassette Transporters
P-Glycoprotein
28 Citations (Scopus)

Endogenous dopamine (DA) competes with the binding of a radiolabeled D3 receptor partial agonist in vivo: A positron emission tomography study

Mach, R. H., Tu, Z., Xu, J., Li, S., Jones, L. A., Taylor, M., Luedtke, R. T., Derdeyn, C. P., Perlmutter, J. S. & Mintun, M. A., 1 Aug 2011, In : Synapse. 65, 8, p. 724-732 9 p.

Research output: Contribution to journalArticleResearchpeer-review

Positron-Emission Tomography
Dopamine
Dopamine D3 Receptors
Lorazepam
Putamen
8 Citations (Scopus)

Evaluation of the D3 dopamine receptor selective agonist/partial agonist PG01042 on l-dopa dependent animal involuntary movements in rats

Riddle, L. R., Kumar, R., Griffin, S. A., Grundt, P., Newman, A. H. & Luedtke, R. T., 1 Feb 2011, In : Neuropharmacology. 60, 2-3, p. 284-294 11 p.

Research output: Contribution to journalArticleResearchpeer-review

Dihydroxyphenylalanine
Dopamine Agonists
Dyskinesias
Adenylyl Cyclases
Dopamine Antagonists
16 Citations (Scopus)

Influence of cocaine history on the behavioral effects of dopamine D 3 receptor-selective compounds in monkeys

Blaylock, B. L., Gould, R. W., Banala, A., Grundt, P., Luedtke, R. T., Newman, A. H. & Nader, M. A., 1 Jan 2011, In : Neuropsychopharmacology. 36, 5, p. 1104-1113 10 p.

Research output: Contribution to journalArticleResearchpeer-review

Cocaine
Haplorhini
Dopamine
History
Quinpirole
49 Citations (Scopus)

N -(3-Fluoro-4-(4-(2-methoxy or 2,3-dichlorophenyl)piperazine-1-yl)butyl) arylcarboxamides as selective dopamine D3 receptor ligands: Critical role of the carboxamide linker for d3 receptor selectivity

Banala, A. K., Levy, B. A., Khatri, S. S., Furman, C. A., Roof, R. A., Mishra, Y., Griffin, S. A., Sibley, D. R., Luedtke, R. T. & Newman, A. H., 26 May 2011, In : Journal of Medicinal Chemistry. 54, 10, p. 3581-3594 14 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Amides
Ligands
Dopamine D2 Receptors
Structure-Activity Relationship
26 Citations (Scopus)

Synthesis and characterization of selective dopamine D 2 receptor ligands using aripiprazole as the lead compound

Vangveravong, S., Zhang, Z., Taylor, M., Bearden, M., Xu, J., Cui, J., Wang, W., Luedtke, R. T. & MacH, R. H., 1 Jun 2011, In : Bioorganic and Medicinal Chemistry. 19, 11, p. 3502-3511 10 p.

Research output: Contribution to journalArticleResearchpeer-review

Benperidol
Domperidone
Lead compounds
Oxalates
Dopamine Antagonists
14 Citations (Scopus)

Synthesis and in vitro biological evaluation of carbonyl group-containing analogues for σ1 receptors

Wang, W., Cui, J., Lu, X., Padakanti, P. K., Xu, J., Parsons, S. M., Luedtke, R. T., Rath, N. P. & Tu, Z., 11 Aug 2011, In : Journal of Medicinal Chemistry. 54, 15, p. 5362-5372 11 p.

Research output: Contribution to journalArticleResearchpeer-review

Vesicular Acetylcholine Transport Proteins
Fluorine
Carbon
Ligands
In Vitro Techniques
27 Citations (Scopus)

Synthesis and pharmacological evaluation of fluorine-containing D 3 dopamine receptor ligands

Tu, Z., Li, S., Cui, J., Xu, J., Taylor, M., Ho, D., Luedtke, R. T. & MacH, R. H., 24 Mar 2011, In : Journal of Medicinal Chemistry. 54, 6, p. 1555-1564 10 p.

Research output: Contribution to journalArticleResearchpeer-review

Fluorine
Dopamine Receptors
Dopamine D4 Receptors
Pharmacology
Dopamine D3 Receptors
2010
27 Citations (Scopus)

[3H]4-(dimethylamino)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)- butyl)benzamide: A selective radioligand for dopamine D3 receptors. II. Quantitative analysis of dopamine D3 and D2 receptor density ratio in the caudate-putamen

Xu, J., Hassanzadeh, B., Chu, W., Tu, Z., Jones, L. A., Luedtke, R. T., Perlmutter, J. S., Mintun, M. A. & Mach, R. H., 1 Jun 2010, In : Synapse. 64, 6, p. 449-459 11 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Dopamine D2 Receptors
Putamen
Raclopride
Macaca mulatta
15 Citations (Scopus)

Dopamine D3 receptor selective ligands with varying intrinsic efficacies at adenylyl cyclase inhibition and mitogenic signaling pathways

Taylor, M., Grundt, P., Griffin, S. A., Newman, A. H. & Luedtke, R. T., 1 Mar 2010, In : Synapse. 64, 3, p. 251-266 16 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Adenylyl Cyclases
Ligands
Amides
Carbon
47 Citations (Scopus)

Subtype selectivity of dopamine receptor ligands: Insights from structure and ligand-based methods

Wang, Q., MacH, R. H., Luedtke, R. T. & Reichert, D. E., 22 Nov 2010, In : Journal of Chemical Information and Modeling. 50, 11, p. 1970-1985 16 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine Receptors
Ligands
interaction
activity structure
predictive model
20 Citations (Scopus)

Synthesis and characterization of selective dopamine D 2 receptor antagonists. 2. Azaindole, benzofuran, and benzothiophene analogs of L-741,626

Vangveravong, S., Taylor, M., Xu, J., Cui, J., Calvin, W., Babic, S., Luedtke, R. T. & MacH, R. H., 15 Jul 2010, In : Bioorganic and Medicinal Chemistry. 18, 14, p. 5291-5300 10 p.

Research output: Contribution to journalArticleResearchpeer-review

Benperidol
Dopamine
Dopamine Antagonists
Dopamine Receptors
Haloperidol
45 Citations (Scopus)

The tetrahydroisoquinoline derivative SB269,652 is an allosteric antagonist at dopamine D3 and D2 receptors

Silvano, E., Millan, M. J., La Cour, C. M., Han, Y., Duan, L., Griffin, S. A., Luedtke, R. T., Aloisi, G., Rossi, M., Zazzeroni, F., Javitch, J. A. & Maggio, R., 1 Nov 2010, In : Molecular Pharmacology. 78, 5, p. 925-934 10 p.

Research output: Contribution to journalArticleResearchpeer-review

Dopamine D3 Receptors
Tetrahydroisoquinolines
Dopamine D2 Receptors
Dopamine
Phosphorylation